PDB entry 6mbo
View 6mbo on RCSB PDB site
Description: GLP Methyltransferase with Inhibitor EML741-P212121 Crystal Form
Class: transferase/transferase inhibitor
Keywords: Histone, H3, Methylation Inhibition, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2018-08-30, released
2019-02-27
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-01-01, with a file datestamp of
2019-12-27.
Experiment type: XRAY
Resolution: 1.59 Å
R-factor: N/A
AEROSPACI score: 0.44
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Histone-lysine N-methyltransferase EHMT1
Species: Homo sapiens [TaxId:9606]
Gene: EHMT1, EUHMTASE1, GLP, KIAA1876, KMT1D
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6mboa_ - Chain 'B':
Compound: Histone-lysine N-methyltransferase EHMT1
Species: Homo sapiens [TaxId:9606]
Gene: EHMT1, EUHMTASE1, GLP, KIAA1876, KMT1D
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6mbob_ - Heterogens: JDG, ZN, SAH, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>6mboA (A:)
verivsrdiargyeripipcvnavdsepcpsnykyvsqncvtspmnidrnithlqycvci
ddcsssncmcgqlsmrcwydkdgrllpefnmaepplifecnhacscwrncrnrvvqnglr
arlqlyrtrdmgwgvrslqdippgtfvceyvgelisdseadvreedsylfdldnkdgevy
cidarfygnvsrfinhhcepnlvpvrvfmahqdlrfpriaffstrlieageqlgfdyger
fwdikgklfscrcgspkcrhs
- Chain 'B':
Sequence, based on SEQRES records: (download)
>6mboB (B:)
verivsrdiargyeripipcvnavdsepcpsnykyvsqncvtspmnidrnithlqycvci
ddcsssncmcgqlsmrcwydkdgrllpefnmaepplifecnhacscwrncrnrvvqnglr
arlqlyrtrdmgwgvrslqdippgtfvceyvgelisdseadvreedsylfdldnkdgevy
cidarfygnvsrfinhhcepnlvpvrvfmahqdlrfpriaffstrlieageqlgfdyger
fwdikgklfscrcgspkcrhs
Sequence, based on observed residues (ATOM records): (download)
>6mboB (B:)
erivsrdiargyeripipcvnavdsepcpsnykyvsqncvtspmnidrnithlqycvcid
dcsssncmcgqlsmrcwydkdgrllpefnmaepplifecnhacscwrncrnrvvqnglra
rlqlyrtrdmgwgvrslqdippgtfvceyvgelisdseadvreedsylfdldngevycid
arfygnvsrfinhhcepnlvpvrvfmahqdlrfpriaffstrlieageqlgfdygerfwd
ikgklfscrcgspkcrhs