PDB entry 6jx4
View 6jx4 on RCSB PDB site
Description: Crystal structure of EGFR 696-1022 T790M in complex with AZD9291 prepared by soaking
Class: transferase
Keywords: Complex, Inhibitor, EGFR., ONCOPROTEIN, TRANSFERASE
Deposited on
2019-04-22, released
2020-04-22
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-11-04, with a file datestamp of
2020-10-30.
Experiment type: XRAY
Resolution: 2.53 Å
R-factor: N/A
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6jx4a_ - Heterogens: YY3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6jx4A (A:)
gamggeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreat
spkankeildeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigs
qyllnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyha
eggkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekge
rlpqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlps
ptdsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>6jx4A (A:)
geapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatspka
nkeildeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigsqyll
nwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekvpikwmal
esilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidv
ymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpsptdsnfyralmd
eedmddvvdadeyli