PDB entry 6jqr

View 6jqr on RCSB PDB site
Description: crystal structure of flt3 in complex with gilteritinib
Deposited on 2019-04-01, released 2019-11-20
The last revision was dated 2019-11-20, with a file datestamp of 2019-11-15.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: N/A
AEROSPACI score: 0.27 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Receptor-type tyrosine-protein kinase FLT3,Receptor-type tyrosine-protein kinase FLT3
    Species: HOMO SAPIENS, synthetic [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
  • Heterogens: C6F, SO4, GOL, CXS, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >6jqrA (A:)
    ryesqlqmvqvtgssdneyfyvdfreyeydlkwefprenlefgkvlgsgafgkvmnatay
    gisktgvsiqvavkmlkekadsserealmselkmmtqlgshenivnllgactlsgpiyli
    feyccygdllnylrskrekfsedeieyenqkrleeeedlnvltfedllcfayqvakgmef
    lefkscvhrdlaarnvlvthgkvvkicdfglardimsdsnyvvrgnarlpvkwmapeslf
    egiytiksdvwsygillweifslgvnpypgipvdanfykliqngfkmdqpfyateeiyii
    mqscwafdsrkrpsfpnltsflgcqladae
    

    Sequence, based on observed residues (ATOM records):
    >6jqrA (A:)
    ryesqlqmvqvtgssdneyfyvdfreyeydlkwefprenlefgkvlgsgafgkvmnatay
    gisvsiqvavkmlkedsserealmselkmmtqlgshenivnllgactlsgpiylifeycc
    ygdllnylrskrekfsnvltfedllcfayqvakgmeflefkscvhrdlaarnvlvthgkv
    vkicdfmsdsnyvvrgnarlpvkwmapeslfegiytiksdvwsygillweifslgvnpyp
    gipvdanfykliqngfkmdqpfyateeiyiimqscwafdsrkrpsfpnltsflgcqlada
    e