PDB entry 6frf
View 6frf on RCSB PDB site
Description: Crystal structure of CREBBP bromodomain complexd with PA10
Class: transferase
Keywords: Inhibitor, Bromodomain, Transferase
Deposited on
2018-02-15, released
2018-08-29
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-10-10, with a file datestamp of
2018-10-05.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: N/A
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: creb-binding protein
Species: Homo sapiens [TaxId:9606]
Gene: CREBBP, CBP
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6frfa1, d6frfa2 - Chain 'B':
Compound: creb-binding protein
Species: Homo sapiens [TaxId:9606]
Gene: CREBBP, CBP
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6frfb_ - Chain 'C':
Compound: creb-binding protein
Species: Homo sapiens [TaxId:9606]
Gene: CREBBP, CBP
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6frfc_ - Chain 'D':
Compound: creb-binding protein
Species: Homo sapiens [TaxId:9606]
Gene: CREBBP, CBP
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6frfd_ - Heterogens: E3T, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6frfA (A:)
smrkkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlsti
krkldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>6frfA (A:)
mrkkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstik
rkldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
- Chain 'B':
Sequence, based on SEQRES records: (download)
>6frfB (B:)
smrkkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlsti
krkldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>6frfB (B:)
ifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrkld
tgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
- Chain 'C':
Sequence, based on SEQRES records: (download)
>6frfC (C:)
smrkkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlsti
krkldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>6frfC (C:)
ifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrkld
tgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqsl
- Chain 'D':
Sequence, based on SEQRES records: (download)
>6frfD (D:)
smrkkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlsti
krkldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>6frfD (D:)
ifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrkld
tgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg