PDB entry 6fcf

View 6fcf on RCSB PDB site
Description: chk1 kinase in complex with compound 44
Class: transferase
Keywords: inhibitor, complex, chk1, kinase, transferase
Deposited on 2017-12-20, released 2018-01-17
The last revision prior to the SCOPe 2.08 freeze date was dated 2018-02-21, with a file datestamp of 2018-02-16.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: N/A
AEROSPACI score: 0.35 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Serine/threonine-protein kinase Chk1
    Species: Homo sapiens [TaxId:9606]
    Gene: CHEK1, CHK1
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d6fcfa_
  • Heterogens: D58, SO4, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6fcfA (A:)
    mavpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicink
    mlnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvy
    lhgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellk
    rrefhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsapla
    llhkilvenpsaritipdikkdrwynkplkkgakrp
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fcfA (A:)
    wdlvqtlgegaygevqlavnrvteeavavkivdmnikkeicinkmlnhenvvkfyghrre
    gniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrdikpenl
    llderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvdvwscgi
    vltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenpsariti
    pdikkdrwynkpl