PDB entry 6ekd
View 6ekd on RCSB PDB site
Description: Crystal structure of JNK3 in complex with a pyridinylimidazole inhibitor
Class: transferase
Keywords: Protein Kinase Activity Map Kinase Activity ATP Binding Protein Phosphorylation, TRANSFERASE
Deposited on
2017-09-26, released
2018-08-08
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-08-22, with a file datestamp of
2018-08-17.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: N/A
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 10
Species: Homo sapiens [TaxId:9606]
Gene: MAPK10, JNK3, JNK3A, PRKM10, SAPK1B
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6ekda_ - Heterogens: B9K, BME, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6ekdA (A:)
ggsmskskvdnqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikkl
srpfqnqthakrayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcq
viqmeldhermsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartag
tsfmmtpyvvtryyrapevilgmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkv
ieqlgtpcpefmkklqptvrnyvenrpkyagltfpklfpdslfpadsehnklkasqardl
lskmlvidpakrisvddalqhpyinvwydpaeveapppqiydkqlderehtieewkeliy
kevmnse
Sequence, based on observed residues (ATOM records): (download)
>6ekdA (A:)
nqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikklsrpfqnqtha
krayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviqmeldher
msyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglvtryyrapevilgmg
ykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieqlgtpcpefmkklqptvrnyve
nrpkyagltfpklfpdslfpadsehnklkasqardllskmlvidpakrisvddalqhpyi
nvwydderehtieewkeliykevmn