PDB entry 6d0f

View 6d0f on RCSB PDB site
Description: Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant in Complex with 3OHTPE and GRIP Peptide
Class: nuclear protein
Keywords: Breast Cancer, Estrogen Receptor, Agonist, NUCLEAR PROTEIN
Deposited on 2018-04-10, released 2019-04-17
The last revision prior to the SCOPe 2.08 freeze date was dated 2020-02-26, with a file datestamp of 2020-02-21.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: N/A
AEROSPACI score: 0.21 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Estrogen receptor
    Species: Homo sapiens [TaxId:9606]
    Gene: ESR1, ESR, NR3A1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P03372
      • engineered mutation (232)
    Domains in SCOPe 2.08: d6d0fa_
  • Chain 'B':
    Compound: Estrogen receptor
    Species: Homo sapiens [TaxId:9606]
    Gene: ESR1, ESR, NR3A1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P03372
      • engineered mutation (232)
    Domains in SCOPe 2.08: d6d0fb_
  • Chain 'C':
    Compound: GRIP peptide
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
    • PDB 6D0F (Start-9)
  • Chain 'D':
    Compound: GRIP peptide
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
    • PDB 6D0F (0-9)
  • Heterogens: FYS, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6d0fA (A:)
    slalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrv
    pgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmvei
    fdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvldkitd
    tlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplsdllleml
    dahrlhapts
    

    Sequence, based on observed residues (ATOM records): (download)
    >6d0fA (A:)
    ltadqmvsalldaeppilyseasmmglltnladrelvhminwakrvpgfvdltlhdqvhl
    lecawleilmiglvwrsmehpgkllfapnllldrnqgmveifdmllatssrfrmmnlqge
    efvclksiillnsgvytleekdhihrvldkitdtlihlmakagltlqqqhqrlaqlllil
    shirhmsnkgmehlysmksdlllemldah
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >6d0fB (B:)
    slalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrv
    pgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmvei
    fdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvldkitd
    tlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplsdllleml
    dahrlhapts
    

    Sequence, based on observed residues (ATOM records): (download)
    >6d0fB (B:)
    alsltadqmvsalldaeppilysefseasmmglltnladrelvhminwakrvpgfvdltl
    hdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvmveifdmllatssr
    frmmnlqgeefvclksiillnsgvytfdhihrvldkitdtlihlmakagltlqqqhqrla
    qlllilshirhmsnkgmehlysmkplsdlllemldah
    

  • Chain 'C':
    No sequence available.

  • Chain 'D':
    No sequence available.