PDB entry 6czw
View 6czw on RCSB PDB site
Description: Crystal structure of PT1940 bound to HIF2a-B*:ARNT-B* complex
Class: transcription
Keywords: Hif2a, Pas B domain, ARNT, hypoxia inducible factor, EPAS1, TRANSCRIPTION
Deposited on
2018-04-09, released
2018-10-31
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-10-31, with a file datestamp of
2018-10-26.
Experiment type: XRAY
Resolution: 1.6 Å
R-factor: N/A
AEROSPACI score: 0.44
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Endothelial PAS domain-containing protein 1
Species: Homo sapiens [TaxId:9606]
Gene: EPAS1, BHLHE73, HIF2A, MOP2, PASD2
Database cross-references and differences (RAF-indexed):
- Uniprot Q99814 (5-End)
- expression tag (2-4)
- engineered mutation (13)
Domains in SCOPe 2.08: d6czwa1, d6czwa2 - Chain 'B':
Compound: Aryl hydrocarbon receptor nuclear translocator
Species: Homo sapiens [TaxId:9606]
Gene: ARNT, BHLHE2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6czwb_ - Heterogens: FO7, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6czwA (A:)
gefkgldsktflsehsmdmkftycddriteligyhpeellgrsayefyhaldsenmtksh
qnlctkgqvvsgqyrmlakhggyvwletqgtviynprnlqpqcimcvnyvlseiekn
Sequence, based on observed residues (ATOM records): (download)
>6czwA (A:)
fkgldsktflsehsmdmkftycddriteligyhpeellgrsayefyhaldsenmtkshqn
lctkgqvvsgqyrmlakhggyvwletqgtviynppqcimcvnyvlseie
- Chain 'B':
Sequence, based on SEQRES records: (download)
>6czwB (B:)
gefkglnvcqptrfisrhniegiftfvdhrcvatvgyqpqellgknivefchpedqqllr
dsfqqvvklkgqvlsvmfrfrsknqewlwmrtssftfqnpysdeieyiictntnvknssq
e
Sequence, based on observed residues (ATOM records): (download)
>6czwB (B:)
cqptrfisrhniegiftfvdhrcvatvgyqpqellgknivefchpedqqllrdsfqqvvk
lkgqvlsvmfrfrsknqewlwmrtssftfqnpysdeieyiictntnvkns