PDB entry 6bsk
View 6bsk on RCSB PDB site
Description: Human PIM1 kinase in complex with compound 12b
Class: TRANSFERASE/TRANSFERASE Inhibitor
Keywords: Kinase, PIM1, inhibitor, TRANSFERASE, TRANSFERASE-TRANSFERASE Inhibitor complex
Deposited on
2017-12-03, released
2018-03-21
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-04-25, with a file datestamp of
2018-04-20.
Experiment type: XRAY
Resolution: 2.57 Å
R-factor: N/A
AEROSPACI score: 0.2
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase pim-1
Species: Homo sapiens [TaxId:9606]
Gene: PIM1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6bska_ - Heterogens: EDO, MVG, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6bskA (A:)
ekeplesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpme
vvllkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffw
qvleavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysp
pewiryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirw
clalrpsdrptfeeiqnhpwmqdvllpqetaeihlh
Sequence, based on observed residues (ATOM records): (download)
>6bskA (A:)
plesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvl
lkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvl
eavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppew
iryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwcla
lrpsdrptfeeiqnhpwmqdvllpqetaeihlh