PDB entry 6aom
View 6aom on RCSB PDB site
Description: Structure of molecular chaperone Grp94 bound to selective inhibitor methyl 2-[2-(2-benzylphenyl)ethyl]-3-chloro-4,6-dihydroxybenzoate
Class: chaperone/inhibitor
Keywords: Grp94, Hsp90, chaperone-inhibitor complex
Deposited on
2017-08-16, released
2017-10-11
The last revision prior to the SCOPe 2.07 freeze date was dated
2017-11-22, with a file datestamp of
2017-11-17.
Experiment type: XRAY
Resolution: 2.87 Å
R-factor: N/A
AEROSPACI score: 0.15
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Endoplasmin
Species: Canis lupus familiaris [TaxId:9615]
Gene: HSP90B1, GRP94, TRA1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d6aoma_ - Chain 'B':
Compound: Endoplasmin
Species: Canis lupus familiaris [TaxId:9615]
Gene: HSP90B1, GRP94, TRA1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d6aomb_ - Heterogens: P33, VC5, GOL, PEG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6aomA (A:)
slreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltdenala
gneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqedgqs
tseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrgtti
tlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktggggktvwdwelmn
Sequence, based on observed residues (ATOM records): (download)
>6aomA (A:)
ekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltdenalagneelt
vkikcdkeknllhvtdtgvgmtreelvknlgtiaktseflnkmtestseligqfgvgfys
aflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrgttitlvlkeeasdylel
dtiknlvkkysqfinfpiyvwsskttvwdwelmn
- Chain 'B':
Sequence, based on SEQRES records: (download)
>6aomB (B:)
slreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltdenala
gneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqedgqs
tseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrgtti
tlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktggggktvwdwelmn
Sequence, based on observed residues (ATOM records): (download)
>6aomB (B:)
ekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltdenalagneelt
vkikcdkeknllhvtdtgvgmtreelvknlgtitseflnkmtestseligqfgvgfysaf
lvadkvivtskhnndtqhiwesdsnefsviadprgntlgrgttitlvlkeeasdyleldt
iknlvkkysqfinfpiyvwssktktvwdwelmn