PDB entry 6acb
View 6acb on RCSB PDB site
Description: Crystal structure of PDE5 in complex with inhibitor LW1805
Class: hydrolase/hydrolase inhibitor
Keywords: PDE5 in complex with inhibitor LW1805, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2018-07-26, released
2018-09-19
The last revision prior to the SCOPe 2.07 freeze date was dated
2018-09-19, with a file datestamp of
2018-09-14.
Experiment type: XRAY
Resolution: 2.8 Å
R-factor: N/A
AEROSPACI score: 0.16
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cGMP-specific 3',5'-cyclic phosphodiesterase
Species: Homo sapiens [TaxId:9606]
Gene: PDE5A, PDE5
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d6acba_ - Heterogens: SO4, ZN, MG, 9T9, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6acbA (A:)
eetrelqslaaavvpsaqtlkitdfsfsdfelsdletalctirmftdlnlvqnfqmkhev
lcrwilsvkknyrknvayhnwrhafntaqcmfaalkagkiqnkltdleilalliaalshd
ldhrgvnnsyiqrsehplaqlychsimehhhfdqclmilnspgnqilsglsieeykttlk
iikqailatdlalyikrrgeffelirknqfnledphqkelflamlmtacdlsaitkpwpi
qqriaelvateffdqgdrerkelnieptdlmnrekknkipsmqvgfidaiclqlyealth
vsedcfplldgcrknrqkwqalaeqq
Sequence, based on observed residues (ATOM records): (download)
>6acbA (A:)
eetrelqslaaavvpsaqtlkitdfsfsdfelsdletalctirmftdlnlvqnfqmkhev
lcrwilsvkknyrknvayhnwrhafntaqcmfaalkagkiqnkltdleilalliaalshd
ldhrgvnnsyiqrsehplaqlychsimehhhfdqclmilnspgnqilsglsieeykttlk
iikqailatdlalyikrrgeffelirknqfnledphqkelflamlmtacdlsaitkpwpi
qqriaelvateffdqekknkipsmqvgfidaiclqlyealthvsedcfplldgcrknrqk
wqalaeqq