PDB entry 5zto
View 5zto on RCSB PDB site
Description: Crystal structure of EGFR 696-1022 T790M/C797S in complex with D3003
Class: transferase
Keywords: EGFR, T790M/C797S, inhibitor, TRANSFERASE
Deposited on
2018-05-04, released
2019-06-12
The last revision prior to the SCOPe 2.08 freeze date was dated
2019-06-12, with a file datestamp of
2019-06-07.
Experiment type: XRAY
Resolution: 2.65 Å
R-factor: N/A
AEROSPACI score: 0.18
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
- Uniprot P00533
- engineered mutation (98)
- engineered mutation (105)
Domains in SCOPe 2.08: d5ztoa_ - Heterogens: 9JO, CL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5ztoA (A:)
gamggeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreat
spkankeildeayvmasvdnphvcrllgicltstvqlimqlmpfgslldyvrehkdnigs
qyllnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyha
eggkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekge
rlpqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlps
ptdsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>5ztoA (A:)
eapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelatspkanke
ildeayvmasvdnphvcrllgicltstvqlimqlmpfgslldyvrehkdnigsqyllnwc
vqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglapikwmalesilhriythqs
dvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidvymimvkcwmida
dsrpkfreliiefskmardpqrylviqgdermhlpsptdsnfymddvvdadeyl