PDB entry 5yqo
View 5yqo on RCSB PDB site
Description: Crystal structure of Sirt2 in complex with selective inhibitor L5C
Class: hydrolase/hydrolase inhibitor
Keywords: NAD-dependent deacetylase sirtuin-2, Inhibitor, Complex, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2017-11-07, released
2018-10-17
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-10-17, with a file datestamp of
2018-10-12.
Experiment type: XRAY
Resolution: 1.48 Å
R-factor: N/A
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: nad-dependent protein deacetylase sirtuin-2
Species: Homo sapiens [TaxId:9606]
Gene: SIRT2, SIR2L, SIR2L2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5yqoa1, d5yqoa2 - Heterogens: ZN, L5C, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5yqoA (A:)
gasgserlldeltlegvarymqsercrrviclvgagistsagipdfrspstglydnleky
hlpypeaifeisyfkkhpepffalakelypgqfkptichyfmrllkdkglllrcytqnid
tleriagleqedlveahgtfytshcvsascrheyplswmkekifsevtpkcedcqslvkp
divffgeslparffscmqsdflkvdlllvmgtslqvqpfasliskaplstprllinkeka
gqsdpflgmimglgggmdfdskkayrdvawlgecdqgclalaellgwkkeledlvrreha
sidaqs
Sequence, based on observed residues (ATOM records): (download)
>5yqoA (A:)
gasgserlldeltlegvarymqsercrrviclvgagistsagipdfrspstpypeaifei
syfkkhpepffalakelypgqfkptichyfmrllkdkglllrcytqnidtleriagleqe
dlveahgtfytshcvsascrheyplswmkekifsevtpkcedcqslvkpdivffgeslpa
rffscmqsdflkvdlllvmgtslqvqpfasliskaplstprllinkekagqsdpflggmd
fdskkayrdvawlgecdqgclalaellgwkkeledlvrrehasidaqs