PDB entry 5ya5
View 5ya5 on RCSB PDB site
Description: CRYSTAL STRUCTURE OF c-MET IN COMPLEX WITH NOVEL INHIBITOR
Class: transferase/inhibitor
Keywords: c-MET inhibitor, TRANSFERASE-INHIBITOR complex
Deposited on
2017-08-30, released
2018-07-04
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-07-04, with a file datestamp of
2018-06-29.
Experiment type: XRAY
Resolution: 1.89 Å
R-factor: N/A
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5ya5a_ - Heterogens: 6TD, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5ya5A (A:)
mgsshhhhhhgdsdisspllqntvhidlsalnpelvqavqhvvigpsslivhfnevigrg
hfgcvyhgtlldndgkkihcavkslnritdigevsqfltegiimkdfshpnvlsllgicl
rsegsplvvlpymkhgdlrnfirnethnptvkdligfglqvakgmkylaskkfvhrdlaa
rncmldekftvkvadfglardmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvw
sfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemr
psfselvsrisaifstfig
Sequence, based on observed residues (ATOM records): (download)
>5ya5A (A:)
alnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtllkkihcavkslnrsqflte
giimkdfshpnvlsllgicsplvvlpymkhgdlrnfirnethnptvkdligfglqvakgm
kylaskkfvhrdlaarncmldekftvkvadfglardmydkeyysvhnktgaklpvkwmal
eslqtqkfttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdpl
yevmlkcwhpkaemrpsfselvsrisaifstfi