PDB entry 5y5t
View 5y5t on RCSB PDB site
Description: Crystal structures of spleen tyrosine kinase in complex with a novel inhibitor
Class: transferase/transferase inhibitor
Keywords: Inhibitor, Spleen Tyrosine Kinase, human kinase, drug discovery, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2017-08-09, released
2018-06-27
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-07-11, with a file datestamp of
2018-07-06.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: N/A
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Tyrosine-protein kinase SYK
Species: Homo sapiens [TaxId:9606]
Gene: SYK
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5y5ta_ - Heterogens: 8OR, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5y5tA (A:)
maleeirpkevyldrklltledkelgsgnfgtvkkgyyqmkkvvktvavkilkneandpa
lkdellaeanvmqqldnpyivrmigiceaeswmlvmemaelgplnkylqqnrhvkdknii
elvhqvsmgmkyleesnfvhrdlaarnvllvtqhyakisdfglskalradenyykaqthg
kwpvkwyapecinyykfssksdvwsfgvlmweafsygqkpyrgmkgsevtamlekgermg
cpagcpremydlmnlcwtydvenrpgfaavelrlrnyyydvvnlehhhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>5y5tA (A:)
vyldrklltledkelgtvkkgyyqmkkvvktvavkilknalkdellaeanvmqqldnpyi
vrmigiceaeswmlvmemaelgplnkylqqnrhvkdkniielvhqvsmgmkyleesnfvh
rdlaarnvllvtqhyakisdfglskalradenyykaqthgkwpvkwyapecinyykfssk
sdvwsfgvlmweafsygqkpyrgmkgsevtamlekgermgcpagcpremydlmnlcwtyd
venrpgfaavelrlrnyyydvvn