PDB entry 5xmx

View 5xmx on RCSB PDB site
Description: Co-crystal structure of Inhibitor compound in complex with human PPARdelta LBD
Class: transcription/inhibitor
Keywords: PPARdelta, Inhibitor compound, TRANSCRIPTION-INHIBITOR complex
Deposited on 2017-05-16, released 2018-05-23
The last revision prior to the SCOPe 2.08 freeze date was dated 2018-05-23, with a file datestamp of 2018-05-18.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Peroxisome proliferator-activated receptor delta
    Species: Homo sapiens [TaxId:9606]
    Gene: PPARD, NR1C2, PPARB
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5xmxa_
  • Chain 'B':
    Compound: Peroxisome proliferator-activated receptor delta
    Species: Homo sapiens [TaxId:9606]
    Gene: PPARD, NR1C2, PPARB
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5xmxb_
  • Heterogens: 89L, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5xmxA (A:)
    gshmqvadlkafskhiynaylknfnmtkkkarsiltgkashtapfvihdietlwqaekgl
    vwkqlvnglppykeisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygv
    heaifamlasivnkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnaleldds
    dlalfiaaiilcgdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadl
    rqlvtehaqmmqrikktetetslhpllqeiykdmy
    

    Sequence, based on observed residues (ATOM records): (download)
    >5xmxA (A:)
    vadlkafskhiynaylknfnmtkkkarsiltgapfvihdietlwqaekglvwglppykei
    svhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygvheaifamlasivnkd
    gllvangsgfvtreflrslrkpfsdiiepkfefavkfnalelddsdlalfiaaiilcgdr
    pglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadlrqlvtehaqmmqrik
    ktetetslhpllqeiyk
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >5xmxB (B:)
    gshmqvadlkafskhiynaylknfnmtkkkarsiltgkashtapfvihdietlwqaekgl
    vwkqlvnglppykeisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygv
    heaifamlasivnkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnaleldds
    dlalfiaaiilcgdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadl
    rqlvtehaqmmqrikktetetslhpllqeiykdmy
    

    Sequence, based on observed residues (ATOM records): (download)
    >5xmxB (B:)
    kafskhiynaylknfnmtkkkarsiltapfvihdietlwqaelppykeisvhvfyrcqct
    tvetvreltefaksipsfsslflndqvtllkygvheaifamlasivnkdgllvangsgfv
    treflrslrkpfsdiiepkfefavkfnalelddsdlalfiaaiilcgdrpglmnvprvea
    iqdtilralefhlqanhpdaqylfpkllqkmadlrqlvtehaqmmqrikktetetslhpl
    lqeiy