PDB entry 5xmx
View 5xmx on RCSB PDB site
Description: Co-crystal structure of Inhibitor compound in complex with human PPARdelta LBD
Class: transcription/inhibitor
Keywords: PPARdelta, Inhibitor compound, TRANSCRIPTION-INHIBITOR complex
Deposited on
2017-05-16, released
2018-05-23
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-05-23, with a file datestamp of
2018-05-18.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Peroxisome proliferator-activated receptor delta
Species: Homo sapiens [TaxId:9606]
Gene: PPARD, NR1C2, PPARB
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5xmxa_ - Chain 'B':
Compound: Peroxisome proliferator-activated receptor delta
Species: Homo sapiens [TaxId:9606]
Gene: PPARD, NR1C2, PPARB
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5xmxb_ - Heterogens: 89L, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5xmxA (A:)
gshmqvadlkafskhiynaylknfnmtkkkarsiltgkashtapfvihdietlwqaekgl
vwkqlvnglppykeisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygv
heaifamlasivnkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnaleldds
dlalfiaaiilcgdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadl
rqlvtehaqmmqrikktetetslhpllqeiykdmy
Sequence, based on observed residues (ATOM records): (download)
>5xmxA (A:)
vadlkafskhiynaylknfnmtkkkarsiltgapfvihdietlwqaekglvwglppykei
svhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygvheaifamlasivnkd
gllvangsgfvtreflrslrkpfsdiiepkfefavkfnalelddsdlalfiaaiilcgdr
pglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadlrqlvtehaqmmqrik
ktetetslhpllqeiyk
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5xmxB (B:)
gshmqvadlkafskhiynaylknfnmtkkkarsiltgkashtapfvihdietlwqaekgl
vwkqlvnglppykeisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygv
heaifamlasivnkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnaleldds
dlalfiaaiilcgdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadl
rqlvtehaqmmqrikktetetslhpllqeiykdmy
Sequence, based on observed residues (ATOM records): (download)
>5xmxB (B:)
kafskhiynaylknfnmtkkkarsiltapfvihdietlwqaelppykeisvhvfyrcqct
tvetvreltefaksipsfsslflndqvtllkygvheaifamlasivnkdgllvangsgfv
treflrslrkpfsdiiepkfefavkfnalelddsdlalfiaaiilcgdrpglmnvprvea
iqdtilralefhlqanhpdaqylfpkllqkmadlrqlvtehaqmmqrikktetetslhpl
lqeiy