PDB entry 5xdl
View 5xdl on RCSB PDB site
Description: Crystal structure of EGFR 696-1022 L858R in complex with CO-1686
Class: transferase
Keywords: EGFR, L858R, inhibitor, TRANSFERASE
Deposited on
2017-03-28, released
2017-12-13
The last revision prior to the SCOPe 2.06 freeze date was dated
2017-12-13, with a file datestamp of
2017-12-08.
Experiment type: XRAY
Resolution: 2.7 Å
R-factor: N/A
AEROSPACI score: 0.18
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
- Uniprot P00533 (4-End)
- engineered mutation (166)
Domains in SCOPe 2.06: d5xdla_ - Heterogens: 8JC, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5xdlA (A:)
gstsgeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreat
spkankeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigs
qyllnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgrakllgaeekeyha
eggkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekge
rlpqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlps
ptdsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>5xdlA (A:)
geapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikeeatspkank
eildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyllnw
cvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgraklpikwmalesilhriyt
hqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidvymimvkcwm
idadsrpkfreliiefskmardpqrylviqgdermhlpedmddvvdadeyli