PDB entry 5ut3
View 5ut3 on RCSB PDB site
Description: JAK2 JH2 in complex with IKK-2 Inhibitor VI
Class: transferase/transferase inhibitor
Keywords: Pseudokinase Domain, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2017-02-14, released
2017-06-07
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-01-01, with a file datestamp of
2019-12-27.
Experiment type: XRAY
Resolution: 1.5 Å
R-factor: N/A
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Tyrosine-protein kinase JAK2
Species: Homo sapiens [TaxId:9606]
Gene: JAK2
Database cross-references and differences (RAF-indexed):
- Uniprot O60674
- engineered mutation (123)
- engineered mutation (241)
- engineered mutation (258)
Domains in SCOPe 2.08: d5ut3a_ - Heterogens: IK1, GOL, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5ut3A (A:)
vfhkirnedlifneslgqgtftkifkgvrrevgdygqlhetevllkvldkahrnysesff
eaasmmsklshkhlvlnygvcvcgdenilvqefvkfgsldtylkknkncinilwklevak
qlaaamhfleentlihgnvcaknillireedrktgnppfiklsdpgisitvlpkdilqer
ipwvppecienpknlnlatdkwsfgttlweicsggdkplsaldsqrklqfyedrhqlpap
kaaelanlinncmdyepdhrpsfraiirdlnslftpdlvprgshhhhhh
Sequence, based on observed residues (ATOM records): (download)
>5ut3A (A:)
fhkirnedlifneslgqgtftkifkgvrrevgdygqlhetevllkvldkahrnysesffe
aasmmsklshkhlvlnygvcvcgdenilvqefvkfgsldtylkknkncinilwklevakq
laaamhfleentlihgnvcaknillireedrktgnppfiklsdpgisitvlpkdilqeri
pwvppecienpknlnlatdkwsfgttlweicsggdkplsaldsqrklqfyedrhqlpapk
aaelanlinncmdyepdhrpsfraiirdlnsl