PDB entry 5upu

View 5upu on RCSB PDB site
Description: Crystal Structure of the Catalytic Domain of the Inosine Monophosphate Dehydrogenase from Mycobacterium tuberculosis in the presence of TBK6
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: IMPDH, delta CBS, Structural Genomics, Center for Structural Genomics of Infectious Diseases, CSGID, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on 2017-02-04, released 2017-02-22
The last revision prior to the SCOPe 2.08 freeze date was dated 2020-01-01, with a file datestamp of 2019-12-27.
Experiment type: XRAY
Resolution: 2.91 Å
R-factor: N/A
AEROSPACI score: 0.15 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: inosine-5'-monophosphate dehydrogenase
    Species: Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) [TaxId:83332]
    Gene: guaB, guaB2, Rv3411c, MTCY78.17
    Database cross-references and differences (RAF-indexed):
    • Uniprot P9WKI7 (Start-127)
      • linker (128-132)
    • Uniprot P9WKI7 (133-End)
    Domains in SCOPe 2.08: d5upua_
  • Heterogens: IMP, 6Q9, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5upuA (A:)
    snamsrgmsgledssdlvvspyvrmgglttdpvptggddphkvamlgltfddvlllpaas
    dvvpatadtssqltkkirlkvplvssamdtvtesrmaiamaraggmgvlhrnlpvaeqag
    qvemvkrsggllvgaavgvggdawvrammlvdagvdvlvvdtahahnrlvldmvgklkse
    vgdrvevvggnvatrsaaaalvdagadavkvgvgpgsicttrvvagvgapqitaileava
    acrpagvpviadgglqysgdiakalaagastamlgsllagtaeapgelifvngkqyksyr
    gmgslgamrgrggatsyskdryfaddalsedklvpegiegrvpfrgplssvihqltgglr
    aamgytgsptievlqqaqfvritpaglkeshphdvamtveapnyyar
    

    Sequence, based on observed residues (ATOM records): (download)
    >5upuA (A:)
    dpvptggddphkvamlgltfddvlllpaasdvvpatadtssqltkkirlkvplvssamdt
    vtesrmaiamaraggmgvlhrnlpvaeqagqvemvkrsggllvgaavgvggdawvramml
    vdagvdvlvvdtahahnrlvldmvgklksevgdrvevvggnvatrsaaaalvdagadavk
    vgvgpgsicttrvvagvgapqitaileavaacrpagvpviadgglqysgdiakalaagas
    tamlgsllagtaeapgelifvngkqyksyrgmgslgamvpegiegrvpfrgplssvihql
    tgglraamgytgsptievlqqaqfvritpagl