PDB entry 5tiu
View 5tiu on RCSB PDB site
Description: Crystal structure of SYK kinase domain with inhibitor
Class: Transferase/Transferase Inhibitor
Keywords: Carboxamide Spleen Tyrosine Kinase (Syk), Transferase-Transferase Inhibitor complex
Deposited on
2016-10-03, released
2017-01-11
The last revision prior to the SCOPe 2.07 freeze date was dated
2017-01-11, with a file datestamp of
2017-01-06.
Experiment type: XRAY
Resolution: 1.49 Å
R-factor: N/A
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Tyrosine-protein kinase SYK
Species: Homo sapiens [TaxId:9606]
Gene: SYK
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d5tiua1, d5tiua2 - Heterogens: 7CU, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5tiuA (A:)
maleeirpkevyldrklltledkelgsgnfgtvkkgyyqmkkvvktvavkilkneandpa
lkdellaeanvmqqldnpyivrmigiceaeswmlvmemaelgplnkylqqnrhvkdknii
elvhqvsmgmkyleesnfvhrdlaarnvllvtqhyakisdfglskalradenyykaqthg
kwpvkwyapecinyykfssksdvwsfgvlmweafsygqkpyrgmkgsevtamlekgermg
cpagcpremydlmnlcwtydvenrpgfaavelrlrnyyydvvneghhhhhh
Sequence, based on observed residues (ATOM records): (download)
>5tiuA (A:)
vyldrklltledkelgtvkkgyyqmkkvvktvavkilkalkdellaeanvmqqldnpyiv
rmigiceaeswmlvmemaelgplnkylqqnrhvkdkniielvhqvsmgmkyleesnfvhr
dlaarnvllvtqhyakisdfglskalradenyykaqthgkwpvkwyapecinyykfssks
dvwsfgvlmweafsygqkpyrgmkgsevtamlekgermgcpagcpremydlmnlcwtydv
enrpgfaavelrlrnyyydvvneghh