PDB entry 5tco
View 5tco on RCSB PDB site
Description: Human p38 MAP Kinase in Complex with Dibenzosuberone Compound 1
Class: transferase
Keywords: Inhibitor, Dibenzosuberone, Human p38 MAP Kinase, transferase
Deposited on
2016-09-15, released
2017-04-19
The last revision prior to the SCOPe 2.06 freeze date was dated
2017-04-19, with a file datestamp of
2017-04-14.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: N/A
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2, SAPK2A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d5tcoa_ - Heterogens: 79Q, BOG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5tcoA (A:)
gsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>5tcoA (A:)
ptfyrqelnktiwevperyqnlspvgssvcaafdtktglrvavkklsrpfqsiihakrty
relrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltddhvqf
liyqilrglkyihsadiihrdlkpsnlavnedcelkildfgltrwyrapeimlnwmhynq
tvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqsl
tqmpkmnfanganplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpydq
sfesrdllidewksltydevisfvppp