PDB entry 5qtf

View 5qtf on RCSB PDB site
Description: T. brucei FPPS in complex with CID 144539
Class: Transferase/Transferase inhibitor
Keywords: farnesyl diphosphate synthase, Trypanosoma brucei, PanDDA, protein-ligand complex, Transferase-Transferase inhibitor complex
Deposited on 2019-08-09, released 2020-10-07
The last revision prior to the SCOPe 2.08 freeze date was dated 2020-10-07, with a file datestamp of 2020-10-02.
Experiment type: XRAY
Resolution: 1.78 Å
R-factor: N/A
AEROSPACI score: 0.46 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: farnesyl pyrophosphate synthase
    Species: Trypanosoma brucei [TaxId:5691]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5qtfa_
  • Heterogens: PK7, PO4, NA, GOL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5qtfA (A:)
    gpmpmqmfmqvydeiqmflleelelkfdmdpnrvrylrkmmdttclggkynrgltvidva
    esllslspnnngeeddgarrkrvlhdacvcgwmieflqahylveddimdnsvtrrgkpcw
    yrhpdvtvqcaindglllkswthmmamhffadrpflqdllcrfnrvdyttavgqlydvts
    mfdsnkldpdvsqptttdfaeftlsnykrivkyktayytyllplvmglivsealptvdmg
    vteelamlmgeyfqvqddvmdcftpperlgkvgtdiqdakcswlavtflakassaqvaef
    kanygsgdsekvatvrrlyeeadlqgdyvayeaavaeqvkelieklrlcspgfaasvetl
    wgktykrqk
    

    Sequence, based on observed residues (ATOM records): (download)
    >5qtfA (A:)
    mpmqmfmqvydeiqmflleelelkfdmdpnrvrylrkmmdttclggkynrgltvidvaes
    llslsgarrkrvlhdacvcgwmieflqahylveddimdnshpdvtvqcaindglllkswt
    hmmamhffadrpflqdllcrfnrvdyttavgqlydvtsmfdsndfaeftlsnykrivkyk
    tayytyllplvmglivsealptvdmgvteelamlmgeyfqvqddvmdcftpperlgkvgt
    diqdakcswlavtflakassaqvaefkanygsgdsekvatvrrlyeeadlqgdyvayeaa
    vaeqvkelieklrlcspgfaasvetlwgkt