PDB entry 5qim
View 5qim on RCSB PDB site
Description: tgf-beta receptor type 1 kinase domain (t204d) in complex with n-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b] pyridin-2-yl]pyridin-2-yl}acetamide
Class: transferase/transferase inhibitor
Keywords: alk5, sb431542, kinase domain, transferase-transferase inhibitor complex, transferase
Deposited on
2018-08-05, released
2018-10-31
The last revision prior to the SCOPe 2.08 freeze date was dated
2021-05-12, with a file datestamp of
2021-05-07.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: N/A
AEROSPACI score: 0.47
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: TGF-beta receptor type-1
Species: Homo sapiens [TaxId:9606]
Gene: TGFBR1, ALK5, SKR4
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5qima1, d5qima2 - Heterogens: J2Y, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5qimA (A:)
ggtiartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhe
nilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlh
meivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtkr
ymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdps
veemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsq
qegikm
Sequence, based on observed residues (ATOM records): (download)
>5qimA (A:)
ggtiartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhe
nilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlh
meivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtkr
ymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdps
veemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsq
qegi