PDB entry 5qil
View 5qil on RCSB PDB site
Description: tgf-beta receptor type 1 kinase domain (t204d) in complex with n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide
Class: transferase/transferase inhibitor
Keywords: alk5, sb431542, kinase domain, transferase-transferase inhibitor complex, transferase
Deposited on
2018-08-05, released
2018-10-31
The last revision prior to the SCOPe 2.07 freeze date was dated
2018-10-31, with a file datestamp of
2018-10-26.
Experiment type: XRAY
Resolution: 1.98 Å
R-factor: N/A
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: TGF-beta receptor type-1
Species: Homo sapiens [TaxId:9606]
Gene: TGFBR1, ALK5, SKR4
Database cross-references and differences (RAF-indexed):
- Uniprot P36897 (3-End)
- expression tag (0-2)
- engineered mutation (7)
Domains in SCOPe 2.07: d5qila1, d5qila2 - Heterogens: J2V, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5qilA (A:)
ghmtiardivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrh
enilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahl
hmeivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtk
rymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdp
sveemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqls
qqegikm
Sequence, based on observed residues (ATOM records): (download)
>5qilA (A:)
ghmtiardivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrh
enilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahl
hmeivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtk
rymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdp
sveemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqls
qqe