PDB entry 5p9m

View 5p9m on RCSB PDB site
Description: btk1 binds covalently to hy-15771 ono-4059
Class: transferase
Keywords: kinase, kinase-ligand complex, TRANSFERASE
Deposited on 2016-09-20, released 2017-05-24
The last revision prior to the SCOPe 2.08 freeze date was dated 2018-02-21, with a file datestamp of 2018-02-16.
Experiment type: XRAY
Resolution: 1.41 Å
R-factor: N/A
AEROSPACI score: 0.53 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Tyrosine-protein kinase BTK
    Species: Homo sapiens [TaxId:9606]
    Gene: BTK, AGMX1, ATK, BPK
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5p9ma_
  • Heterogens: 7GB, DMS, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5p9mA (A:)
    gknapstaglgygsweidpkdltflkelgtgqfgvvkygkwrgqydvaikmikegsmsed
    efieeakvmmnlsheklvqlygvctkqrpifiiteymangcllnylremrhrfqtqqlle
    mckdvceameyleskqflhrdlaarnclvndqgvvkvsdfglsryvlddeytssvgskfp
    vrwsppevlmyskfssksdiwafgvlmweiyslgkmpyerftnsetaehiaqglrlyrph
    lasekvytimyscwhekaderptfkillsnildvmdees
    

    Sequence, based on observed residues (ATOM records): (download)
    >5p9mA (A:)
    glgygsweidpkdltflkelgtgqfgvvkygkwrgqydvaikmikegsmsedefieeakv
    mmnlsheklvqlygvctkqrpifiiteymangcllnylremrhrfqtqqllemckdvcea
    meyleskqflhrdlaarnclvndqgvvkvsdfglsryvlddeytssvgskfpvrwsppev
    lmyskfssksdiwafgvlmweiyslgkmpyerftnsetaehiaqglrlyrphlasekvyt
    imyscwhekaderptfkillsnildvmdees