PDB entry 5ox5

View 5ox5 on RCSB PDB site
Description: HIF prolyl hydroxylase 2 (PHD2/ EGLN1) in complex with CCT6, a GSK1278863-related compound
Class: oxidoreductase
Keywords: oxidoreductase, non-heme dioxygenase, iron, 2-oxoglutarate, hypoxia-inducible factor, hif, hif prolyl hydroxylase domain 2, phd2, egln1, oxygenase, hypoxia, DNA-binding, metal-binding, transcription, helix-loop-helix-beta, dsbh, facial triad, cytoplasm, transcription/epigenetic regulation, signaling, development, cell structure, beta-hydroxylation, transcription activator/inhibitor, ubl conjugation, polymorphism, vitamin c, zinc-finger, familial erythrocytosis, breast cancer, transcription complex
Deposited on 2017-09-06, released 2017-10-18
The last revision prior to the SCOPe 2.08 freeze date was dated 2018-02-21, with a file datestamp of 2018-02-16.
Experiment type: XRAY
Resolution: 2.25 Å
R-factor: N/A
AEROSPACI score: 0.25 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Egl nine homolog 1
    Species: Homo sapiens [TaxId:9606]
    Gene: EGLN1, C1orf12, PNAS-118, PNAS-137
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5ox5a_
  • Heterogens: MN, B2E, BCT, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5ox5A (A:)
    gshmaspngqtkplpalklaleyivpcmnkhgicvvddflgketgqqigdevralhdtgk
    ftdgqlvsqksdsskdirgdkitwiegkepgcetigllmssmddlirhcngklgsyking
    rtkamvacypgngtgyvrhvdnpngdgrcvtciyylnkdwdakvsggilrifpegkaqfa
    diepkfdrllffwsdrrnphevqpayatryaitvwyfdaderarakvkyltgekgvrvel
    nkpsdsvgkdvf
    

    Sequence, based on observed residues (ATOM records): (download)
    >5ox5A (A:)
    lpalklaleyivpcmnkhgicvvddflgketgqqigdevralhdtgkftdgqlvsqksds
    skdirgdkitwiegkepgcetigllmssmddlirhcngklgsykingrtkamvacypgng
    tgyvrhvdnpngdgrcvtciyylnkdwdakvsggilrifpegkaqfadiepkfdrllffw
    sdrrnphevqpayatryaitvwyfdaderarakvkyvrvel