PDB entry 5o8v
View 5o8v on RCSB PDB site
Description: Covalent Inhibitor 4a bound to the Lipid Pocket of p38alpha Mutant S251C
Class: transferase
Keywords: kinase, small molecule, lipid pocket, p38, covalent, mutant, TRANSFERASE
Deposited on
2017-06-14, released
2017-09-06
The last revision prior to the SCOPe 2.06 freeze date was dated
2017-09-06, with a file datestamp of
2017-09-01.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2, SAPK2A
Database cross-references and differences (RAF-indexed):
- Uniprot Q16539
- engineered mutation (250)
Domains in SCOPe 2.06: d5o8va_ - Heterogens: 9O2, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5o8vA (A:)
msqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkicsesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>5o8vA (A:)
rptfyrqelnktiwevperyqnlspvgsgsvcaafdtktglrvavkklsrpfqsiihakr
tyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnniltddhvqfliy
qilrglkyihsadiihrdlkpsnlavnedcelkildvatrwyrapeimlnwmhynqtvdi
wsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkicsesarnyiqsltqmp
kmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpydqs
fesrdllidewksltydevisfvpppld