PDB entry 5ngf

View 5ngf on RCSB PDB site
Description: Crystal structure of USP7 in complex with the covalent inhibitor, FT827
Class: hydrolase
Keywords: Deubiquitination, Hydrolase
Deposited on 2017-03-17, released 2017-10-18
The last revision prior to the SCOPe 2.06 freeze date was dated 2017-10-25, with a file datestamp of 2017-10-20.
Experiment type: XRAY
Resolution: 2.33 Å
R-factor: N/A
AEROSPACI score: 0.24 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Ubiquitin carboxyl-terminal hydrolase 7
    Species: Homo sapiens [TaxId:9606]
    Gene: USP7, HAUSP
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.06: d5ngfa_
  • Chain 'B':
    Compound: Ubiquitin carboxyl-terminal hydrolase 7
    Species: Homo sapiens [TaxId:9606]
    Gene: USP7, HAUSP
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.06: d5ngfb_
  • Heterogens: 8WN, EDO, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5ngfA (A:)
    gskkhtgyvglknqgatcymnsllqtlfftnqlrkavymmptegddssksvplalqrvfy
    elqhsdkpvgtkkltksfgwetldsfmqhdvqelcrvlldnvenkmkgtcvegtipklfr
    gkmvsyiqckevdyrsdrredyydiqlsikgkknifesfvdyvaveqldgdnkydagehg
    lqeaekgvkfltlppvlhlqlmrfmydpqtdqnikindrfefpeqlpldeflqktdpkdp
    anyilhavlvhsgdnhgghyvvylnpkgdgkwckfdddvvsrctkeeaiehnygghdddl
    svrhctnaymlvyiresklsevlqavtdhdipqqlverlqeekrieaqkrkerqe
    

    Sequence, based on observed residues (ATOM records): (download)
    >5ngfA (A:)
    khtgyvglknqgatcymnsllqtlfftnqlrkavymmptegddssksvplalqrvfyelq
    hsdkpvgtkkltksfgwetldsfmqhdvqelcrvlldnvenkmkgtcvegtipklfrgkm
    vsyiqckevdyrsdrredyydiqlsikgkknifesfvdyvaveqldgdnkydagehglqe
    aekgvkfltlppvlhlqlmrfmynikindrfefpeqlpldeflqktdpkdpanyilhavl
    vhsgdnhgghyvvylnpkgdgkwckfdddvvsrctkeeaiehnygghctnaymlvyires
    klsevlqavtdhdipqqlverlqeekrieaqk
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >5ngfB (B:)
    gskkhtgyvglknqgatcymnsllqtlfftnqlrkavymmptegddssksvplalqrvfy
    elqhsdkpvgtkkltksfgwetldsfmqhdvqelcrvlldnvenkmkgtcvegtipklfr
    gkmvsyiqckevdyrsdrredyydiqlsikgkknifesfvdyvaveqldgdnkydagehg
    lqeaekgvkfltlppvlhlqlmrfmydpqtdqnikindrfefpeqlpldeflqktdpkdp
    anyilhavlvhsgdnhgghyvvylnpkgdgkwckfdddvvsrctkeeaiehnygghdddl
    svrhctnaymlvyiresklsevlqavtdhdipqqlverlqeekrieaqkrkerqe
    

    Sequence, based on observed residues (ATOM records): (download)
    >5ngfB (B:)
    khtgyvglknqgatcymnsllqtlfftnqlrkavymmptegddssksvplalqrvfyelq
    hsdkpvgtkkltksfgwetldsfmqhdvqelcrvlldnvenkmkgtcvegtipklfrgkm
    vsyiqckevdyrsdrredyydiqlsikgkknifesfvdyvaveqldgdnkydagehglqe
    aekgvkfltlppvlhlqlmrfmynikindrfefpeqlpldeflqktdpkdpanyilhavl
    vhsgdnhgghyvvylnpkgdgkwckfdddvvsrctkeeaiehnygghctnaymlvyires
    klsevlqavtdhdipqqlverlqeekrieaqk