PDB entry 5n9n
View 5n9n on RCSB PDB site
Description: Crystal structure of human Protein kinase CK2 catalytic subunit in complex with the ATP-competitive, tight-binding dibenzofuran inhibitor TF85 (4a)
Class: transferase
Keywords: Protein kinase, CK2, Casein kinase 2, Protein phosphorylation, ATP-competitive inhititors, dibenzofuran derivatives, transferase, TIGHT-BINDING INHIBITORS
Deposited on
2017-02-25, released
2018-02-28
The last revision prior to the SCOPe 2.07 freeze date was dated
2018-03-07, with a file datestamp of
2018-03-02.
Experiment type: XRAY
Resolution: 1.84 Å
R-factor: N/A
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Casein kinase II subunit alpha
Species: Homo sapiens [TaxId:9606]
Gene: CSNK2A1, CK2A1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d5n9na_ - Heterogens: 8QK, ACT, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5n9nA (A:)
msgpvpsrarvytdvnthrpreywdyeshvvewgnqddyqlvrklgrgkysevfeainit
nnekvvvkilkpvkkkkikreikilenlrggpniitladivkdpvsrtpalvfehvnntd
fkqlyqtltdydirfymyeilkaldychsmgimhrdvkphnvmidhehrklrlidwglae
fyhpgqeynvrvasryfkgpellvdyqmydysldmwslgcmlasmifrkepffhghdnyd
qlvriakvlgtedlydyidkynieldprfndilgrhsrkrwerfvhsenqhlvspealdf
ldkllrydhqsrltareamehpyfytvvkdqarmg
Sequence, based on observed residues (ATOM records): (download)
>5n9nA (A:)
sgpvpsrarvytdvnthrpreywdyeshvvewgnqddyqlvrklgrgkysevfeainitn
nekvvvkilkpvkkkkikreikilenlrggpniitladivkdpvsrtpalvfehvnntdf
kqlyqtltdydirfymyeilkaldychsmgimhrdvkphnvmidhehrklrlidwglaef
yhpgqeynvrvasryfkgpellvdyqmydysldmwslgcmlasmifrkepffhghdnydq
lvriakvlgtedlydyidkynieldprfndilgrhsrkrwerfvhsenqhlvspealdfl
dkllrydhqsrltareamehpyfytvvkd