PDB entry 5mqy
View 5mqy on RCSB PDB site
Description: CATHEPSIN L IN COMPLEX WITH 4-[1,3-benzodioxol-5-ylmethyl(2-phenoxyethyl)amino]-5-fluoropyrimidine-2-carbonitrile
Class: hydrolase
Keywords: protease inhibitor, hydrolase-hydrolase inhibitor complex, hydrolase
Deposited on
2016-12-21, released
2017-03-22
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-06-07, with a file datestamp of
2017-06-02.
Experiment type: XRAY
Resolution: 1.13 Å
R-factor: N/A
AEROSPACI score: 0.7
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Cathepsin L1
Species: Homo sapiens [TaxId:9606]
Gene: CTSL, CTSL1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5mqya_ - Heterogens: GH4, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5mqyA (A:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfestesdnn
kywlvknswgeewgmggyvkmakdrrnhcgiasaasyptv
Sequence, based on observed residues (ATOM records): (download)
>5mqyA (A:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfestnkywl
vknswgeewgmggyvkmakdrrnhcgiasaasyptv