PDB entry 5mfv

View 5mfv on RCSB PDB site
Description: Crystal structure of the GluK1 ligand-binding domain in complex with kainate and BPAM-521 at 2.18 A resolution
Class: membrane protein
Keywords: ionotropic glutamate receptor, GluK1 ligand-binding domain, membrane protein, positive allosteric modulator
Deposited on 2016-11-18, released 2017-04-12
The last revision prior to the SCOPe 2.08 freeze date was dated 2018-01-17, with a file datestamp of 2018-01-12.
Experiment type: XRAY
Resolution: 2.18 Å
R-factor: N/A
AEROSPACI score: 0.27 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Grik1, Glur5
    Database cross-references and differences (RAF-indexed):
    • Uniprot P22756 (Start-115)
      • see remark 999 (33)
      • linker (116-117)
    • Uniprot P22756 (118-End)
    Domains in SCOPe 2.08: d5mfva_
  • Chain 'B':
    Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Grik1, Glur5
    Database cross-references and differences (RAF-indexed):
    • Uniprot P22756 (Start-115)
      • see remark 999 (33)
      • linker (116-117)
    • Uniprot P22756 (118-256)
    Domains in SCOPe 2.08: d5mfvb_
  • Heterogens: 5PX, KAI, CL, SO4, GOL, ACT, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5mfvA (A:)
    ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
    ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
    dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
    lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
    gklhmmkekwwrgngcp
    

    Sequence, based on observed residues (ATOM records): (download)
    >5mfvA (A:)
    rtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkyga
    qndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsa
    ddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvltt
    dyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegkl
    hmmkekwwrg
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >5mfvB (B:)
    ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
    ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
    dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
    lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
    gklhmmkekwwrgngcp
    

    Sequence, based on observed residues (ATOM records): (download)
    >5mfvB (B:)
    tlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkygaq
    ngewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsaddl
    akqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvlttdya
    llmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegklhmm
    kekwwrgngcp