PDB entry 5m2v
View 5m2v on RCSB PDB site
Description: Structure of GluK1 ligand-binding domain (S1S2) in complex with (2S,4R)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid at 3.18 A resolution
Class: membrane protein
Keywords: Kainate receptor ligand-binding domain, GluK1-LBD, GluK1-S1S2, antagonist, membrane protein
Deposited on
2016-10-13, released
2017-01-11
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-08-09, with a file datestamp of
2017-08-04.
Experiment type: XRAY
Resolution: 3.18 Å
R-factor: N/A
AEROSPACI score: 0.12
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1, Glur5
Database cross-references and differences (RAF-indexed):
- Uniprot P22756 (Start-115)
- conflict (33)
- linker (116-117)
- Uniprot P22756 (118-256)
Domains in SCOPe 2.08: d5m2va_ - Chain 'B':
Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1, Glur5
Database cross-references and differences (RAF-indexed):
- Uniprot P22756 (Start-115)
- conflict (33)
- linker (116-117)
- Uniprot P22756 (118-256)
Domains in SCOPe 2.08: d5m2vb_ - Heterogens: 7E5, SO4, CL
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5m2vA (A:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp
Sequence, based on observed residues (ATOM records): (download)
>5m2vA (A:)
tlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkygaq
ndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsad
dlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvlttd
yallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegklh
mmkekwwrgcp
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5m2vB (B:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp
Sequence, based on observed residues (ATOM records): (download)
>5m2vB (B:)
tlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkygaq
ndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsad
dlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvlttd
yallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegklh
mmkekwwrgngcp