PDB entry 5laq
View 5laq on RCSB PDB site
Description: Crystal structure of human phosphodiesterase 4B catalytic domain with inhibitor NPD-001
Class: hydrolase
Keywords: Phosphodiesterase, hydrolase, cAMP, alternative splicing
Deposited on
2016-06-14, released
2018-03-14
The last revision prior to the SCOPe 2.07 freeze date was dated
2018-03-14, with a file datestamp of
2018-03-09.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: N/A
AEROSPACI score: 0.23
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP-specific 3',5'-cyclic phosphodiesterase 4B,cAMP-specific 3',5'-cyclic phosphodiesterase 4B
Species: Homo sapiens [TaxId:9606]
Gene: PDE4B, DPDE4
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d5laqa_ - Heterogens: ZN, MG, ACT, 6M5, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5laqA (A:)
msvsemasnkfkrmlnrelthlsemsrsgnqvseyisntfldkqndveipkvtaeeapqp
mtqisgvkklmhssslnntsisrfgvntenedhlakeledlnkwglnifnvagyshnrpl
tcimyaifqerdllktfrissdtfitymmtledhyhsdvayhnslhaadvaqsthvllst
paldavftdleilaaifaaaihdvdhpgvsnqflintnselalmyndesvlenhhlavgf
kllqeehcdifmnltkkqrqtlrkmvidmvlatdmskhmslladlktmvetkkvtssgvl
lldnytdriqvlrnmvhcadlsnptkslelyrqwtdrimeeffqqgdkerergmeispmc
dkhtasveksqvgfidyivhplwetwadlvqpdaqdildtlednrnwyqsmipqshhhhh
h
Sequence, based on observed residues (ATOM records): (download)
>5laqA (A:)
tsisrfgvntenedhlakeledlnkwglnifnvagyshnrpltcimyaifqerdllktfr
issdtfitymmtledhyhsdvayhnslhaadvaqsthvllstpaldavftdleilaaifa
aaihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqeehcdifmnltkkq
rqtlrkmvidmvlatdmskhmslladlktmvetkkvtssgvllldnytdriqvlrnmvhc
adlsnptkslelyrqwtdrimeeffqqgdkerergmeispmcdkhtasveksqvgfidyi
vhplwetwadlvqpdaqdildtlednrnwyqsmipqs