PDB entry 5krt
View 5krt on RCSB PDB site
Description: HIV-1 Integrase Catalytic Core Domain (CCD) in Complex with a Fragment-Derived Allosteric Inhibitor
Class: hydrolase, transferase/inhibitor
Keywords: HIV-1 Integrase; Catalytic Core Domain (CCD); p75/LEDGF inhibitor, hydrolase, transferase-inhibitor complex
Deposited on
2016-07-07, released
2016-09-28
The last revision prior to the SCOPe 2.06 freeze date was dated
2016-09-28, with a file datestamp of
2016-09-23.
Experiment type: XRAY
Resolution: 1.65 Å
R-factor: N/A
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: integrase
Species: Human immunodeficiency virus 1 [TaxId:11676]
Database cross-references and differences (RAF-indexed):
- Uniprot Q76353 (2-152)
- expression tag (1)
- engineered mutation (130)
Domains in SCOPe 2.06: d5krta1, d5krta2 - Heterogens: 6W6, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5krtA (A:)
dsspgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvh
tdngsnftsttvkaacwwagikqefgipynpqsqgviesmnkelkkiigqvrdqaehlkt
avqmavfihnkkrkggiggysagerivdiiatd
Sequence, based on observed residues (ATOM records): (download)
>5krtA (A:)
sspgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvht
dngsnftsttvkaacwwagikqefgipynpgviesmnkelkkiigqvrdqaehlktavqm
avfihnkkrggysagerivdiiatd