PDB entry 5krs
View 5krs on RCSB PDB site
Description: HIV-1 Integrase Catalytic Core Domain in Complex with an Allosteric Inhibitor, 3-(1H-pyrrol-1-yl)-2-thiophenecarboxylic acid
Class: hydrolase, transferase/inhibitor
Keywords: HIV-1 Integrase Catalytic Core Domain, p75/LEDGF inhibitor, hydrolase, transferase-inhibitor complex
Deposited on
2016-07-07, released
2016-09-28
The last revision prior to the SCOPe 2.07 freeze date was dated
2016-11-16, with a file datestamp of
2016-11-11.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: N/A
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: integrase
Species: Human immunodeficiency virus 1 [TaxId:11676]
Database cross-references and differences (RAF-indexed):
- Uniprot Q76353 (2-152)
- expression tag (0-1)
- engineered mutation (130)
Domains in SCOPe 2.07: d5krsa1, d5krsa2 - Heterogens: DMS, 6XI, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5krsA (A:)
dsspgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvh
tdngsnftsttvkaacwwagikqefgipynpqsqgviesmnkelkkiigqvrdqaehlkt
avqmavfihnkkrkggiggysagerivdiiatd
Sequence, based on observed residues (ATOM records): (download)
>5krsA (A:)
dsspgiwqldcthlegkvilvavhvasgyieaevipaetgqetayfllklagrwpvktvh
tdngsnftsttvkaacwwagikqefgipynpgviesmnkelkkiigqvrdqaehlktavq
mavfihnkkrkgggysagerivdiiatd