PDB entry 5k9c
View 5k9c on RCSB PDB site
Description: Crystal structure of human dihydroorotate dehydrogenase with ML390
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: Oxidoreductase, alpha/beta barrel, inhibitor, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2016-05-31, released
2016-10-12
The last revision prior to the SCOPe 2.06 freeze date was dated
2016-10-12, with a file datestamp of
2016-10-07.
Experiment type: XRAY
Resolution: 1.66 Å
R-factor: N/A
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dihydroorotate dehydrogenase (quinone), mitochondrial
Species: Homo sapiens [TaxId:9606]
Gene: DHODH
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d5k9ca_ - Heterogens: FNR, ORO, MLJ, SO4, ACT, CL, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5k9cA (A:)
smatgderfyaehlmptlqglldpesahrlavrftslgllprarfqdsdmlevrvlghkf
rnpvgiaagfdkhgeavdglykmgfgfveigsvtpkpqegnprprvfrlpedqavinryg
fnshglsvvehrlrarqqkqakltedglplgvnlgknktsvdaaedyaegvrvlgplady
lvvnvsspntaglrslqgkaelrrlltkvlqerdglrrvhrpavlvkiapdltsqdkedi
asvvkelgidglivtnttvsrpaglqgalrsetgglsgkplrdlstqtiremyaltqgrv
piigvggvssgqdalekiragaslvqlytaltfwgppvvgkvkreleallkeqgfggvtd
aigadhrr
Sequence, based on observed residues (ATOM records): (download)
>5k9cA (A:)
erfyaehlmptlqglldpesahrlavrftslgllprarfqdsdmlevrvlghkfrnpvgi
aagfdkhgeavdglykmgfgfveigsvtpkpqegnprprvfrlpedqavinrygfnshgl
svvehrlrarqqkqakltedglplgvnlgknktsvdaaedyaegvrvlgpladylvvnvs
spntgkaelrrlltkvlqerdglrrvhrpavlvkiapdltsqdkediasvvkelgidgli
vtnttvsrpaglqgalrsetgglsgkplrdlstqtiremyaltqgrvpiigvggvssgqd
alekiragaslvqlytaltfwgppvvgkvkreleallkeqgfggvtdaigadhrr