PDB entry 5j7g
View 5j7g on RCSB PDB site
Description: Structure of MDM2 with low molecular weight inhibitor with aliphatic linker.
Class: ligase
Keywords: p53, MDM2, MDMX, protein-protein interaction, cancer, inhibitor, ligase
Deposited on
2016-04-06, released
2017-05-17
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-01-31, with a file datestamp of
2018-01-26.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: N/A
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
- Uniprot Q00987 (1-End)
- initiating methionine (0)
Domains in SCOPe 2.08: d5j7ga1, d5j7ga2 - Chain 'B':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
- Uniprot Q00987 (1-End)
- initiating methionine (0)
Domains in SCOPe 2.08: d5j7gb_ - Chain 'C':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
- Uniprot Q00987 (1-End)
- initiating methionine (0)
Domains in SCOPe 2.08: d5j7gc_ - Chain 'D':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
- Uniprot Q00987 (1-End)
- initiating methionine (0)
Domains in SCOPe 2.08: d5j7gd_ - Heterogens: 6GG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5j7gA (A:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqessdsgtsvsen
Sequence, based on observed residues (ATOM records): (download)
>5j7gA (A:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvv
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5j7gB (B:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqessdsgtsvsen
Sequence, based on observed residues (ATOM records): (download)
>5j7gB (B:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqe
- Chain 'C':
Sequence, based on SEQRES records: (download)
>5j7gC (C:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqessdsgtsvsen
Sequence, based on observed residues (ATOM records): (download)
>5j7gC (C:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvn
- Chain 'D':
Sequence, based on SEQRES records: (download)
>5j7gD (D:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqessdsgtsvsen
Sequence, based on observed residues (ATOM records): (download)
>5j7gD (D:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvn