PDB entry 5ia1
View 5ia1 on RCSB PDB site
Description: Crystal Structure of Ephrin A2 (EphA2) Receptor Protein Kinase with MLN8054
Class: transferase
Keywords: transferase, tyrosine-protein kinase, receptor, ATP-binding
Deposited on
2016-02-21, released
2016-11-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2019-06-12, with a file datestamp of
2019-06-07.
Experiment type: XRAY
Resolution: 2.04 Å
R-factor: N/A
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Ephrin type-A receptor 2
Species: Homo sapiens [TaxId:9606]
Gene: EPHA2, ECK
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5ia1a_ - Heterogens: ZZL, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5ia1A (A:)
gdpnqavlkftteihpscvtrqkvigagefgevykgmlktssgkkevpvaiktlkagyte
kqrvdflgeagimgqfshhniirlegviskykpmmiiteymengaldkflrekdgefsvl
qlvgmlrgiaagmkylanmnyvhrdlaarnilvnsnlvckvsdfglsrvleddpeatytt
sggkipirwtapeaisyrkftsasdvwsfgivmwevmtygerpywelsnhevmkaindgf
rlptpmdcpsaiyqlmmqcwqqerarrpkfadivsildklirapdslktladfdprvsir
lpstsg
Sequence, based on observed residues (ATOM records): (download)
>5ia1A (A:)
tteihpscvtrqkvigagefgevykgmlkevpvaiktlkagytekqrvdflgeagimgqf
shhniirlegviskykpmmiiteymengaldkflrekdgefsvlqlvgmlrgiaagmkyl
anmnyvhrdlaarnilvnsnlvckvsdfglsipirwtapeaisyrkftsasdvwsfgivm
wevmtygerpywelsnhevmkaindgfrlptpmdcpsaiyqlmmqcwqqerarrpkfadi
vsildklirapdslktladfd