PDB entry 5h8g

View 5h8g on RCSB PDB site
Description: Crystal structure of CK2 with compound 7b
Class: Transferase/Transferase Inhibitor
Keywords: Kinase, Inhibitor, CK2, Transferase-Transferase Inhibitor complex
Deposited on 2015-12-23, released 2016-02-10
The last revision prior to the SCOPe 2.08 freeze date was dated 2016-03-30, with a file datestamp of 2016-03-25.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Casein kinase II subunit alpha
    Species: Homo sapiens [TaxId:9606]
    Gene: CSNK2A1, CK2A1
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5h8ga_
  • Heterogens: CL, EDO, 5Y4, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5h8gA (A:)
    msgpvpsrarvytdvnthrpreywdyeshvvewgnqddyqlvrklgrgkysevfeainit
    nnekvvvkilkpvkkkkikreikilenlrggpniitladivkdpvsrtpalvfehvnntd
    fkqlyqtltdydirfymyeilkaldychsmgimhrdvkphnvmidhehrklrlidwglae
    fyhpgqeynvrvasryfkgpellvdyqmydysldmwslgcmlasmifrkepffhghdnyd
    qlvriakvlgtedlydyidkynieldprfndilgrhsrkrwerfvhsenqhlvspealdf
    ldkllrydhqsrltareamehpyfytvvkdqar
    

    Sequence, based on observed residues (ATOM records): (download)
    >5h8gA (A:)
    gpvpsrarvytdvnthrpreywdyeshvvewgnqddyqlvrklgrgkysevfeainitnn
    ekvvvkilkkkkkikreikilenlrggpniitladivkdpvsrtpalvfehvnntdfkql
    yqtltdydirfymyeilkaldychsmgimhrdvkphnvmidhehrklrlidwglaefyhp
    gqeynvrvasryfkgpellvdyqmydysldmwslgcmlasmifrkepffhghdnydqlvr
    iakvlgtedlydyidkynieldprfndilgrhsrkrwerfvhsenqhlvspealdfldkl
    lrydhqsrltareamehpyfytvv