PDB entry 5g1z

View 5g1z on RCSB PDB site
Description: Plasmodium vivax N-myristoyltransferase in complex with a quinoline inhibitor (compound 1)
Class: transferase
Keywords: transferase, myristoylation, malaria, inhibitor, quinoline, drug design
Deposited on 2016-04-06, released 2017-02-15
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-06-28, with a file datestamp of 2017-06-23.
Experiment type: XRAY
Resolution: 1.5 Å
R-factor: N/A
AEROSPACI score: 0.48 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glycylpeptide N-tetradecanoyltransferase
    Species: Plasmodium vivax [TaxId:5855]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5g1za1, d5g1za2
  • Chain 'B':
    Compound: Glycylpeptide N-tetradecanoyltransferase
    Species: Plasmodium vivax [TaxId:5855]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5g1zb1, d5g1zb2
  • Chain 'C':
    Compound: Glycylpeptide N-tetradecanoyltransferase
    Species: Plasmodium vivax [TaxId:5855]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5g1zc1, d5g1zc2
  • Heterogens: NHW, U53, DMS, MG, SO4, CL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence; same for both SEQRES and ATOM records: (download)
    >5g1zA (A:)
    idykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrs
    eiytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaip
    tdicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkp
    vsdaryyhrsinvkklieigfsslnsrltmsraiklyrvedtlniknmrlmkkkdvegvh
    kllgsyleqfnlyavftkeeiahwflpienviytyvneengkikdmisfyslpsqilgnd
    kystlnaaysfynvtttatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegd
    gslkyylynwkcasfapahvgivll
    

  • Chain 'B':
    Sequence; same for both SEQRES and ATOM records: (download)
    >5g1zB (B:)
    idykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrs
    eiytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaip
    tdicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkp
    vsdaryyhrsinvkklieigfsslnsrltmsraiklyrvedtlniknmrlmkkkdvegvh
    kllgsyleqfnlyavftkeeiahwflpienviytyvneengkikdmisfyslpsqilgnd
    kystlnaaysfynvtttatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegd
    gslkyylynwkcasfapahvgivll
    

  • Chain 'C':
    Sequence, based on SEQRES records: (download)
    >5g1zC (C:)
    idykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrs
    eiytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaip
    tdicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkp
    vsdaryyhrsinvkklieigfsslnsrltmsraiklyrvedtlniknmrlmkkkdvegvh
    kllgsyleqfnlyavftkeeiahwflpienviytyvneengkikdmisfyslpsqilgnd
    kystlnaaysfynvtttatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegd
    gslkyylynwkcasfapahvgivll
    

    Sequence, based on observed residues (ATOM records): (download)
    >5g1zC (C:)
    dykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrse
    iytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaipt
    dicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkpv
    sdaryyhrsinvkklieigflyrvedtlniknmrlmkkkdvegvhkllgsyleqfnlyav
    ftkeeiahwflpienviytyvneengkikdmisfyslpsqilgndkystlnaaysfynvt
    ttatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegdgslkyylynwkcasf
    apahvgivll