PDB entry 5fpe

View 5fpe on RCSB PDB site
Description: Structure of heat shock-related 70kDA protein 2 with small-molecule ligand 1H-1,2,4-triazol-3-amine (AT485) in an alternate binding site.
Class: chaperone
Keywords: heat shock-related protein, heat shock, chaperone, hsp70, hspa2, protein-ligand complex, fragment screening, alternate binding site, at485.
Deposited on 2015-11-28, released 2015-12-23
The last revision prior to the SCOPe 2.08 freeze date was dated 2016-01-13, with a file datestamp of 2016-01-08.
Experiment type: XRAY
Resolution: 1.96 Å
R-factor: N/A
AEROSPACI score: 0.32 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: heat shock-related 70kda protein 2
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5fpea1, d5fpea2
  • Chain 'B':
    Compound: heat shock-related 70kda protein 2
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5fpeb1, d5fpeb2
  • Heterogens: 3TR, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5fpeA (A:)
    gshmrgpaigidlgttyscvgvfqhgkveiiandqgnrttpsyvaftdterligdaaknq
    vamnptntifdakrligrkfedatvqsdmkhwpfrvvseggkpkvqveykgetktffpee
    issmvltkmkeiaeaylggkvhsavitvpayfndsqrqatkdagtitglnvlriinepta
    aaiaygldkkgcaggeknvlifdlgggtfdvsiltiedgifevkstagdthlggedfdnr
    mvshlaeefkrkhkkdigpnkravrrlrtacerakrtlssstqasieidslyegvdfyts
    itrarfeelnadlfrgtlepvekalrdakldkgqiqeivlvggstripkiqkllqdffng
    kelnksinpdeavaygaavqaailigd
    

    Sequence, based on observed residues (ATOM records): (download)
    >5fpeA (A:)
    gpaigidlgttyscvgvfqhgkveiiandqgnrttpsyvaftdterligdaaknqvamnp
    tntifdakrligrkfedatvqsdmkhwpfrvvseggkpkvqveykgetktffpeeissmv
    ltkmkeiaeaylggkvhsavitvpayfndsqrqatkdagtitglnvlriineptaaaiay
    gldkkggeknvlifdlgggtfdvsiltiedgifevkstagdthlggedfdnrmvshlaee
    fkrkhkkdigpnkravrrlrtacerakrtlssstqasieidslyegvdfytsitrarfee
    lnadlfrgtlepvekalrdakldkgqiqeivlvggstripkiqkllqdffngkelnksin
    pdeavaygaavqaailigd
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >5fpeB (B:)
    gshmrgpaigidlgttyscvgvfqhgkveiiandqgnrttpsyvaftdterligdaaknq
    vamnptntifdakrligrkfedatvqsdmkhwpfrvvseggkpkvqveykgetktffpee
    issmvltkmkeiaeaylggkvhsavitvpayfndsqrqatkdagtitglnvlriinepta
    aaiaygldkkgcaggeknvlifdlgggtfdvsiltiedgifevkstagdthlggedfdnr
    mvshlaeefkrkhkkdigpnkravrrlrtacerakrtlssstqasieidslyegvdfyts
    itrarfeelnadlfrgtlepvekalrdakldkgqiqeivlvggstripkiqkllqdffng
    kelnksinpdeavaygaavqaailigd
    

    Sequence, based on observed residues (ATOM records): (download)
    >5fpeB (B:)
    gpaigidlgttyscvgvfqhgkveiiandqgnrttpsyvaftdterligdaaknqvamnp
    tntifdakrligrkfedatvqsdmkhwpfrvvseggkpkvqveykgetktffpeeissmv
    ltkmkeiaeaylggkvhsavitvpayfndsqrqatkdagtitglnvlriineptaaaiay
    gldkkgcaggeknvlifdlgggtfdvsiltiedgifevkstagdthlggedfdnrmvshl
    aeefkrkhkkdigpnkravrrlrtacerakrtlssstqasieidslyegvdfytsitrar
    feelnadlfrgtlepvekalrdakldkgqiqeivlvggstripkiqkllqdffngkelnk
    sinpdeavaygaavqaailigd