PDB entry 5f2p

View 5f2p on RCSB PDB site
Description: Crystal structure of the BRD9 bromodomain in complex with compound 3.
Class: transcription
Keywords: Bromodomain, Inhibitor, REGULATORY PROTEINS, transcription
Deposited on 2015-12-02, released 2016-03-09
The last revision prior to the SCOPe 2.08 freeze date was dated 2016-06-08, with a file datestamp of 2016-06-03.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: N/A
AEROSPACI score: 0.38 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: brd9
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5f2pa_
  • Chain 'B':
    Compound: brd9
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5f2pb_
  • Heterogens: 5TY, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5f2pA (A:)
    smlklsaenestpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmk
    dkivaneyksvtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkr
    sms
    

    Sequence, based on observed residues (ATOM records): (download)
    >5f2pA (A:)
    stpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmkdkivaneyks
    vtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkrsms
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >5f2pB (B:)
    smlklsaenestpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmk
    dkivaneyksvtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkr
    sms
    

    Sequence, based on observed residues (ATOM records): (download)
    >5f2pB (B:)
    stpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmkdkivaneyks
    vtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkrsms