PDB entry 5ek9

View 5ek9 on RCSB PDB site
Description: Crystal structure of the second bromodomain of human BRD2 in complex with a tetrahydroquinoline inhibitor
Class: transcription
Keywords: chromatin and transcription regulator, acetylation, Structural Genomics, Structural Genomics Consortium, SGC, transcription
Deposited on 2015-11-03, released 2016-11-16
The last revision prior to the SCOPe 2.08 freeze date was dated 2018-01-17, with a file datestamp of 2018-01-12.
Experiment type: XRAY
Resolution: 2.08 Å
R-factor: N/A
AEROSPACI score: 0.3 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Bromodomain-containing protein 2
    Species: Homo sapiens [TaxId:9606]
    Gene: BRD2, KIAA9001, RING3
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5ek9a_
  • Chain 'B':
    Compound: Bromodomain-containing protein 2
    Species: Homo sapiens [TaxId:9606]
    Gene: BRD2, KIAA9001, RING3
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5ek9b_
  • Heterogens: 5P4, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5ek9A (A:)
    smgklseqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkr
    kmenrdyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
    

    Sequence, based on observed residues (ATOM records): (download)
    >5ek9A (A:)
    eqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenrd
    yrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmp
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >5ek9B (B:)
    smgklseqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkr
    kmenrdyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
    

    Sequence, based on observed residues (ATOM records): (download)
    >5ek9B (B:)
    eqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenrd
    yrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmp