PDB entry 5ek9
View 5ek9 on RCSB PDB site
Description: Crystal structure of the second bromodomain of human BRD2 in complex with a tetrahydroquinoline inhibitor
Class: transcription
Keywords: chromatin and transcription regulator, acetylation, Structural Genomics, Structural Genomics Consortium, SGC, transcription
Deposited on
2015-11-03, released
2016-11-16
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-01-17, with a file datestamp of
2018-01-12.
Experiment type: XRAY
Resolution: 2.08 Å
R-factor: N/A
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Gene: BRD2, KIAA9001, RING3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5ek9a_ - Chain 'B':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Gene: BRD2, KIAA9001, RING3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5ek9b_ - Heterogens: 5P4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5ek9A (A:)
smgklseqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkr
kmenrdyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
Sequence, based on observed residues (ATOM records): (download)
>5ek9A (A:)
eqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenrd
yrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmp
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5ek9B (B:)
smgklseqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkr
kmenrdyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
Sequence, based on observed residues (ATOM records): (download)
>5ek9B (B:)
eqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenrd
yrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmp