PDB entry 5e8w
View 5e8w on RCSB PDB site
Description: tgf-beta receptor type 1 kinase domain (t204d) in complex with staurosporine
Class: transferase/transferase inhibitor
Keywords: alk5, kinase domain, transferase-transferase inhibitor complex
Deposited on
2015-10-14, released
2016-05-11
The last revision prior to the SCOPe 2.07 freeze date was dated
2016-05-11, with a file datestamp of
2016-05-06.
Experiment type: XRAY
Resolution: 1.86 Å
R-factor: N/A
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: TGF-beta receptor type-1
Species: Homo sapiens [TaxId:9606]
Gene: TGFBR1, ALK5, SKR4
Database cross-references and differences (RAF-indexed):
- Uniprot P36897 (3-End)
- expression tag (2)
- engineered mutation (7)
Domains in SCOPe 2.07: d5e8wa1, d5e8wa2 - Heterogens: STU, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5e8wA (A:)
ghmtiardivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrh
enilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahl
hmeivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtk
rymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdp
sveemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqls
qqegikm
Sequence, based on observed residues (ATOM records): (download)
>5e8wA (A:)
mtiardivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhen
ilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlhm
eivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtkry
mapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsv
eemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqq
egi