PDB entry 5cau
View 5cau on RCSB PDB site
Description: EGFR kinase domain mutant "TMLR" with compound 41b
Class: Transferase/transferase inhibitor
Keywords: protein kinase inhibitor, Transferase-transferase inhibitor complex
Deposited on
2015-06-29, released
2015-10-28
The last revision prior to the SCOPe 2.06 freeze date was dated
2015-12-02, with a file datestamp of
2015-11-27.
Experiment type: XRAY
Resolution: 2.25 Å
R-factor: N/A
AEROSPACI score: 0.26
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
- Uniprot P00533
- engineered mutation (96)
- engineered mutation (164)
Domains in SCOPe 2.06: d5caua_ - Heterogens: SO4, 4ZR, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5cauA (A:)
gsgeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatsp
kankeildeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigsqy
llnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgrakllgaaaaeyhaeg
gkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerl
pqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpspt
dsnfyralmdeedmddvvdadeylipqqgns
Sequence, based on observed residues (ATOM records): (download)
>5cauA (A:)
geapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelspkankei
ldeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigsqyllnwcv
qiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgraklvpikwmalesilhriyth
qsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidvymimvkcwmi
dadsrpkfreliiefskmardpqrylviqgdermhlpsptdsnfymddvvdadeyli