PDB entry 5a5i

View 5a5i on RCSB PDB site
Description: Cytochrome 2C9 P450 inhibitor complex
Class: oxidoreductase
Keywords: oxidoreductase
Deposited on 2015-06-18, released 2016-08-24
The last revision prior to the SCOPe 2.06 freeze date was dated 2016-08-24, with a file datestamp of 2016-08-18.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.3 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Cytochrome P450 2C9
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
    • Uniprot P11712 (Start-471)
      • expression tag (472-474)
    Domains in SCOPe 2.06: d5a5ia1, d5a5ia2
  • Heterogens: XI1, HEM, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5a5iA (A:)
    makktssgrgklppgptplpvignilqigikdisksltnlskvygpvftlyfglkpivvl
    hgyeavkealidlgeefsgrgifplaeranrgfgivfsngkkwkeirrfslmtlrnfgmg
    krsiedrvqeearclveelrktkaspcdptfilgcapcnvicsiifhkrfdykdqqflnl
    meklnenikilsspwiqicnnfspiidyfpgthnkllknvafmksyilekvkehqesmdm
    nnpqdfidcflmkmekekhnqpseftieslentavdlfgagtettsttlryalllllkhp
    evtakvqeeiervigrnrspcmqdrshmpytdavvhevqryidllptslphavtcdikfr
    nylipkgttilisltsvlhdnkefpnpemfdphhfldeggnfkkskyfmpfsagkricvg
    ealagmelflfltsilqnfnlkslvdpknldttpvvngfasvppfyqlcfipihhhh
    

    Sequence, based on observed residues (ATOM records): (download)
    >5a5iA (A:)
    rgklppgptplplqigikdisksltnlskvygpvftlyfglkpivvlhgyeavkealidl
    geefsgrgilaeranrgfgivfsngkkwkeirrfslmtlrnfgmgkrsiedrvqeearcl
    veelrktkaspcdptfilgcapcnvicsiifhkrfdykdqqflnlmeklnenikilsspw
    ipiidyfpgthnkllknvafmksyilekvkehqesmdmnnpqdfidcflmkmekekhnqp
    seftieslentavdlfgagtettsttlryalllllkhpevtakvqeeiervigrnrspcm
    qdrshmpytdavvhevqryidllptslphavtcdikfrnylipkgttilisltsvlhdnk
    efpnpemfdphhfldeggnfkkskyfmpfsagkricvgealagmelflfltsilqnfnlk
    slvdpknldttpvvngfasvppfyqlcfipihh