PDB entry 4zzz
View 4zzz on RCSB PDB site
Description: Structure of human PARP1 catalytic domain bound to an isoindolinone inhibitor
Class: transferase
Keywords: transferase, human parp1, artd1,
Deposited on
2015-04-15, released
2015-08-12
The last revision prior to the SCOPe 2.07 freeze date was dated
2015-09-23, with a file datestamp of
2015-09-18.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: N/A
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Poly [ADP-ribose] polymerase 1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Chain 'B':
Compound: Poly [ADP-ribose] polymerase 1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d4zzzb1, d4zzzb2 - Heterogens: SO4, GOL, FSU, HOH
PDB Chain Sequences:
- Chain 'A':
No sequence available.
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4zzzB (B:)
gpltvnpgtksklpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysi
lsevqqavsqgssdsqildlsnrfytliphdfgmkkppllnnadsvqakvemldnlldie
vaysllrggsddsskdpidvnyeklktdikvvdrdseeaeiirkyvknthatthnaydle
vidifkieregecqrykpfkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfg
kgiyfadmvsksanychtsqgdpiglillgevalgnmyelkhashisklpkgkhsvkglg
kttpdpsanisldgvdvplgtgissgvndtsllyneyivydiaqvnlkyllklkfnfkts
lw
Sequence, based on observed residues (ATOM records): (download)
>4zzzB (B:)
klpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysilsevqqavsqg
ssdsqildlsnrfytliphdfgmkkppllnnadsvqakvemldnlldievaysllrggdp
idvnyeklktdikvvdrdseeaeiirkyvknthatthnaydlevidifkieregecqryk
pfkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfgkgiyfadmvsksanych
tsqgdpiglillgevalgnmyelkhashisklpkgkhsvkglgkttpdpsanisldgvdv
plgtgissgvndtsllyneyivydiaqvnlkyllklkfnfkt