PDB entry 4zgk
View 4zgk on RCSB PDB site
Description: Structure of Mdm2 with low molecular weight inhibitor.
Class: ligase
Keywords: p53-Mdm2/MdmX interaction, inhibitor, ligase
Deposited on
2015-04-23, released
2016-10-19
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-12-28, with a file datestamp of
2016-12-22.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
- Uniprot Q00987 (1-End)
- initiating methionine (0)
Domains in SCOPe 2.08: d4zgka1, d4zgka2 - Chain 'B':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4zgkb_ - Heterogens: 4NX, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4zgkA (A:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqe
Sequence, based on observed residues (ATOM records): (download)
>4zgkA (A:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvv
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4zgkB (B:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqe
Sequence, based on observed residues (ATOM records): (download)
>4zgkB (B:)
qipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivyc
sndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqqe