PDB entry 4zfi
View 4zfi on RCSB PDB site
Description: Structure of Mdm2 with low molecular weight inhibitor
Class: ligase
Keywords: p53-binding protein Mdm2, Oncoprotein Mdm2, Double minute 2 protein, Hdm2, small molecule inhibitor, ligase
Deposited on
2015-04-21, released
2016-10-19
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-12-28, with a file datestamp of
2016-12-22.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4zfia_ - Chain 'B':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
- Uniprot Q00987 (1-96)
- initiating methionine (0)
Domains in SCOPe 2.08: d4zfib_ - Chain 'C':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4zfic_ - Chain 'D':
Compound: E3 ubiquitin-protein ligase Mdm2
Species: Homo sapiens [TaxId:9606]
Gene: MDM2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4zfid_ - Heterogens: 4NJ, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4zfiA (A:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqq
Sequence, based on observed residues (ATOM records): (download)
>4zfiA (A:)
qipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivyc
sndllgdlfgvpsfsvkehrkiytmiyrnlvvvnq
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>4zfiB (B:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqq
- Chain 'C':
Sequence, based on SEQRES records: (download)
>4zfiC (C:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqq
Sequence, based on observed residues (ATOM records): (download)
>4zfiC (C:)
qipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivyc
sndllgdlfgvpsfsvkehrkiytmiyrnlvvv
- Chain 'D':
Sequence, based on SEQRES records: (download)
>4zfiD (D:)
mqipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivy
csndllgdlfgvpsfsvkehrkiytmiyrnlvvvnqq
Sequence, based on observed residues (ATOM records): (download)
>4zfiD (D:)
ipaseqetlvrpkplllkllksvgaqkdtytmkevlfylgqyimtkrlydekqqhivycs
ndllgdlfgvpsfsvkehrkiytmiyrnlvvvn