PDB entry 4ymb
View 4ymb on RCSB PDB site
Description: Structure of the ligand-binding domain of GluK1 in complex with the antagonist CNG10111
Class: signaling protein
Keywords: Ionotropic glutamate receptor, kainate receptor GluK1, ligand-binding domain, antagonist, signaling protein, fusion protein
Deposited on
2015-03-06, released
2015-08-05
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-08-09, with a file datestamp of
2017-08-04.
Experiment type: XRAY
Resolution: 1.93 Å
R-factor: N/A
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1, Glur5
Database cross-references and differences (RAF-indexed):
- Uniprot P22756 (Start-115)
- variant (33)
- linker (116-117)
- Uniprot P22756 (118-256)
Domains in SCOPe 2.08: d4ymba_ - Chain 'B':
Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1, Glur5
Database cross-references and differences (RAF-indexed):
- Uniprot P22756 (1-115)
- variant (33)
- linker (116-117)
- Uniprot P22756 (118-End)
Domains in SCOPe 2.08: d4ymbb1 - Heterogens: 4E7, ACT, CL, PEG, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4ymbA (A:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp
Sequence, based on observed residues (ATOM records): (download)
>4ymbA (A:)
rtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkyga
qndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsa
ddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvltt
dyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegkl
hmmkekwwrgcp
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4ymbB (B:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp
Sequence, based on observed residues (ATOM records): (download)
>4ymbB (B:)
anrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgky
gaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpid
saddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvl
ttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeeg
klhmmkekwwrgngc