PDB entry 4ymb

View 4ymb on RCSB PDB site
Description: Structure of the ligand-binding domain of GluK1 in complex with the antagonist CNG10111
Class: signaling protein
Keywords: Ionotropic glutamate receptor, kainate receptor GluK1, ligand-binding domain, antagonist, signaling protein, fusion protein
Deposited on 2015-03-06, released 2015-08-05
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-08-09, with a file datestamp of 2017-08-04.
Experiment type: XRAY
Resolution: 1.93 Å
R-factor: N/A
AEROSPACI score: 0.33 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Grik1, Glur5
    Database cross-references and differences (RAF-indexed):
    • Uniprot P22756 (Start-115)
      • variant (33)
      • linker (116-117)
    • Uniprot P22756 (118-256)
    Domains in SCOPe 2.08: d4ymba_
  • Chain 'B':
    Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Grik1, Glur5
    Database cross-references and differences (RAF-indexed):
    • Uniprot P22756 (1-115)
      • variant (33)
      • linker (116-117)
    • Uniprot P22756 (118-End)
    Domains in SCOPe 2.08: d4ymbb1
  • Heterogens: 4E7, ACT, CL, PEG, EDO, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4ymbA (A:)
    ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
    ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
    dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
    lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
    gklhmmkekwwrgngcp
    

    Sequence, based on observed residues (ATOM records): (download)
    >4ymbA (A:)
    rtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkyga
    qndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsa
    ddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvltt
    dyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegkl
    hmmkekwwrgcp
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >4ymbB (B:)
    ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
    ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
    dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
    lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
    gklhmmkekwwrgngcp
    

    Sequence, based on observed residues (ATOM records): (download)
    >4ymbB (B:)
    anrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgky
    gaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpid
    saddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvl
    ttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeeg
    klhmmkekwwrgngc